Gago F - Search Results

1

Double Arylation of the Indole Side Chain of Tri- and Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV-1 and EV-A71 Entry Inhibitors†.

Martí-Marí O, Martínez-Gualda B, de la Puente-Secades S, Mills A, Quesada E, Abdelnabi R, Sun L, Boonen A, Noppen S, Neyts J, Schols D, Camarasa MJ, Gago F, San-Félix A. Martí-Marí O, et al. Among authors: gago f. J Med Chem. 2021 Jul 22;64(14):10027-10046. doi: 10.1021/acs.jmedchem.1c00315. Epub 2021 Jul 7. J Med Chem. 2021. PMID: 34229438 Free PMC article.

2

DNA sequence-specific reading by echinomycin: role of hydrogen bonding and stacking interactions.

Gallego J, Luque FJ, Orozco M, Burgos C, Alvarez-Builla J, Rodrigo MM, Gago F. Gallego J, et al. Among authors: gago f. J Med Chem. 1994 May 27;37(11):1602-9. doi: 10.1021/jm00037a010. J Med Chem. 1994. PMID: 8201593

3

Assessment of solvation effects on calculated binding affinity differences: trypsin inhibition by flavonoids as a model system for congeneric series.

Checa A, Ortiz AR, de Pascual-Teresa B, Gago F. Checa A, et al. Among authors: gago f. J Med Chem. 1997 Dec 5;40(25):4136-45. doi: 10.1021/jm970245v. J Med Chem. 1997. PMID: 9406602

4

Comparative binding energy analysis of HIV-1 protease inhibitors: incorporation of solvent effects and validation as a powerful tool in receptor-based drug design.

Pérez C, Pastor M, Ortiz AR, Gago F. Pérez C, et al. Among authors: gago f. J Med Chem. 1998 Mar 12;41(6):836-52. doi: 10.1021/jm970535b. J Med Chem. 1998. PMID: 9526559

5

Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptase.

Velázquez S, Chamorro C, Pérez-Pérez MJ, Alvarez R, Jimeno ML, Martín-Domenech A, Pérez C, Gago F, De Clercq E, Balzarini J, San-Félix A, Camarasa MJ. Velázquez S, et al. Among authors: gago f. J Med Chem. 1998 Nov 5;41(23):4636-47. doi: 10.1021/jm980370m. J Med Chem. 1998. PMID: 9804703 Free article.

6

Regiospecific synthesis and anti-human immunodeficiency virus activity of novel 5-substituted N-alkylcarbamoyl and N,N-dialkylcarbamoyl 1,2,3-triazole-TSAO analogues.

Velázquez S, Alvarez R, Pérez C, Gago F, De Clercq E, Balzarini J, Camarasa MJ. Velázquez S, et al. Among authors: gago f. Antivir Chem Chemother. 1998 Nov;9(6):481-9. doi: 10.1177/095632029800900604. Antivir Chem Chemother. 1998. PMID: 9865386

7

Novel 3'-spiro nucleoside analogues of TSAO-T. Part II. A comparative study based on NMR conformational analysis in solution and theoretical calculations.

Alvarez R, Jimeno ML, Gago F, Balzarini J, Pérez-Pérez MJ, Camarasa MJ. Alvarez R, et al. Among authors: gago f. Antivir Chem Chemother. 1998 Jul;9(4):333-40. Antivir Chem Chemother. 1998. PMID: 9875412

8

Identification of a putative binding site for [2',5'-bis-O-(tert-butyldimethylsilyl)-beta-D-ribofuranosyl]-3'-spiro-5''-(4''-amino-1'',2''-oxathiole-2'',2''-dioxide)thymine (TSAO) derivatives at the p51-p66 interface of HIV-1 reverse transcriptase.

Rodríguez-Barrios F, Pérez C, Lobatón E, Velázquez S, Chamorro C, San-Félix A, Pérez-Pérez MJ, Camarasa MJ, Pelemans H, Balzarini J, Gago F. Rodríguez-Barrios F, et al. Among authors: gago f. J Med Chem. 2001 Jun 7;44(12):1853-65. doi: 10.1021/jm001095i. J Med Chem. 2001. PMID: 11384232

9

Exploring the role of the 5'-position of TSAO-T. Synthesis and anti-HIV evaluation of novel TSAO-T derivatives.

Chamorro C, Pérez-Pérez MJ, Rodríguez-Barrios F, Gago F, De Clercq E, Balzarini J, San-Félix A, Camarasa MJ. Chamorro C, et al. Among authors: gago f. Antiviral Res. 2001 Jun;50(3):207-22. doi: 10.1016/s0166-3542(01)00145-0. Antiviral Res. 2001. PMID: 11397508

10

Synthesis of 3' '-substituted TSAO derivatives with anti-HIV-1 and anti-HIV-2 activity through an efficient palladium-catalyzed cross-coupling approach.

Lobatón E, Rodríguez-Barrios F, Gago F, Pérez-Pérez MJ, De Clercq E, Balzarini J, Camarasa MJ, Velázquez S. Lobatón E, et al. Among authors: gago f. J Med Chem. 2002 Aug 29;45(18):3934-45. doi: 10.1021/jm020820h. J Med Chem. 2002. PMID: 12190315

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

256 results

Search Page

Filters