Bazureau JP - Search Results

1

Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A.

Bourahla K, Guihéneuf S, Limanton E, Paquin L, Le Guével R, Charlier T, Rahmouni M, Durieu E, Lozach O, Carreaux F, Meijer L, Bazureau JP. Bourahla K, et al. Among authors: bazureau jp. Pharmaceuticals (Basel). 2021 Oct 27;14(11):1086. doi: 10.3390/ph14111086. Pharmaceuticals (Basel). 2021. PMID: 34832868 Free PMC article.

2

Parallel solution-phase synthesis of 2-alkylthio-5-arylidene-3,5-dihydro-4H-imidazol-4-one by one-pot three-component domino reaction.

Renault S, Bertrand S, Carreaux F, Bazureau JP. Renault S, et al. Among authors: bazureau jp. J Comb Chem. 2007 Nov-Dec;9(6):935-42. doi: 10.1021/cc070022i. Epub 2007 Sep 7. J Comb Chem. 2007. PMID: 17822301

3

Reactivity of 2-thiohydantoins towards various electrophilic reagents: applications to the synthesis of new 2-ylidene-3,5-dihydro-4H-imidazol-4-ones.

Chérouvrier JR, Carreaux F, Bazureau JP. Chérouvrier JR, et al. Among authors: bazureau jp. Molecules. 2004 Sep 30;9(10):867-75. doi: 10.3390/91000867. Molecules. 2004. PMID: 18007487 Free PMC article.

4

Synthesis and preliminary biological evaluation of new derivatives of the marine alkaloid leucettamine B as kinase inhibitors.

Debdab M, Renault S, Lozach O, Meijer L, Paquin L, Carreaux F, Bazureau JP. Debdab M, et al. Among authors: bazureau jp. Eur J Med Chem. 2010 Feb;45(2):805-10. doi: 10.1016/j.ejmech.2009.10.009. Epub 2009 Oct 12. Eur J Med Chem. 2010. PMID: 19879673

5

Leucettines, a class of potent inhibitors of cdc2-like kinases and dual specificity, tyrosine phosphorylation regulated kinases derived from the marine sponge leucettamine B: modulation of alternative pre-RNA splicing.

Debdab M, Carreaux F, Renault S, Soundararajan M, Fedorov O, Filippakopoulos P, Lozach O, Babault L, Tahtouh T, Baratte B, Ogawa Y, Hagiwara M, Eisenreich A, Rauch U, Knapp S, Meijer L, Bazureau JP. Debdab M, et al. Among authors: bazureau jp. J Med Chem. 2011 Jun 23;54(12):4172-86. doi: 10.1021/jm200274d. Epub 2011 May 26. J Med Chem. 2011. PMID: 21615147

6

A practical approach to new (5Z) 2-alkylthio-5-arylmethylene-1-methyl-1,5-dihydro-4H-imidazol-4-one derivatives.

Bourahla K, Paquin L, Lozach O, Meijer L, Carreaux F, Bazureau JP. Bourahla K, et al. Among authors: bazureau jp. Molecules. 2011 Aug 30;16(9):7377-90. doi: 10.3390/molecules16097377. Molecules. 2011. PMID: 21878858 Free PMC article.

7

An efficient approach to dispacamide A and its derivatives.

Guihéneuf S, Paquin L, Carreaux F, Durieu E, Meijer L, Bazureau JP. Guihéneuf S, et al. Among authors: bazureau jp. Org Biomol Chem. 2012 Feb 7;10(5):978-87. doi: 10.1039/c1ob06161e. Epub 2011 Dec 8. Org Biomol Chem. 2012. PMID: 22159215

8

Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.

Tahtouh T, Elkins JM, Filippakopoulos P, Soundararajan M, Burgy G, Durieu E, Cochet C, Schmid RS, Lo DC, Delhommel F, Oberholzer AE, Pearl LH, Carreaux F, Bazureau JP, Knapp S, Meijer L. Tahtouh T, et al. Among authors: bazureau jp. J Med Chem. 2012 Nov 8;55(21):9312-30. doi: 10.1021/jm301034u. Epub 2012 Oct 8. J Med Chem. 2012. PMID: 22998443

9

Synthesis of N,N'-bis(5-arylidene-4-oxo-3,5-dihydro-4H-imidazol-2-yl)diamines bearing various linkers and biological evaluation as potential inhibitors of kinases.

Coulibaly WK, Paquin L, Bénie A, Bekro YA, Durieu E, Meijer L, Bazureau JP. Coulibaly WK, et al. Among authors: bazureau jp. Eur J Med Chem. 2012 Dec;58:581-90. doi: 10.1016/j.ejmech.2012.08.044. Epub 2012 Sep 7. Eur J Med Chem. 2012. PMID: 23174317

10

Synthesis of New N,N'-Bis(5-arylidene-4-oxo-4,5-dihydrothiazolin-2-yl)piperazine Derivatives Under Microwave Irradiation and Preliminary Biological Evaluation.

Coulibaly WK, Paquin L, Bénié A, Bekro YA, Durieux E, Meijer L, Le Guével R, Corlu A, Bazureau JP. Coulibaly WK, et al. Among authors: bazureau jp. Sci Pharm. 2012 Oct-Dec;80(4):825-36. doi: 10.3797/scipharm.1206-04. Epub 2012 Sep 16. Sci Pharm. 2012. PMID: 23264934 Free PMC article.

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