Daelemans D - Search Results

1

Inhibition of XPO-1 Mediated Nuclear Export through the Michael-Acceptor Character of Chalcones.

Gargantilla M, López-Fernández J, Camarasa MJ, Persoons L, Daelemans D, Priego EM, Pérez-Pérez MJ. Gargantilla M, et al. Among authors: daelemans d. Pharmaceuticals (Basel). 2021 Nov 6;14(11):1131. doi: 10.3390/ph14111131. Pharmaceuticals (Basel). 2021. PMID: 34832913 Free PMC article.

2

Selective inhibition of Human Immunodeficiency Virus type 1 (HIV-1) by a novel family of tricyclic nucleosides.

Bonache MC, Cordeiro A, Quesada E, Vanstreels E, Daelemans D, Camarasa MJ, Balzarini J, San-Félix A. Bonache MC, et al. Among authors: daelemans d. Antiviral Res. 2011 Oct;92(1):37-44. doi: 10.1016/j.antiviral.2011.05.002. Epub 2011 May 12. Antiviral Res. 2011. PMID: 21600933

3

Synthesis and Biological Evaluation of Pyrrolo[2,1-f][1,2,4]triazine C-Nucleosides with a Ribose, 2'-Deoxyribose, and 2',3'-Dideoxyribose Sugar Moiety.

Li Q, Lescrinier E, Groaz E, Persoons L, Daelemans D, Herdewijn P, De Jonghe S. Li Q, et al. Among authors: daelemans d. ChemMedChem. 2018 Jan 8;13(1):97-104. doi: 10.1002/cmdc.201700657. Epub 2017 Dec 12. ChemMedChem. 2018. PMID: 29160955

4

Design and Synthesis of New 6-Nitro and 6-Amino-3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole Derivatives: Antiproliferative and Antibacterial Activity.

Cuartas V, Crespo MDP, Priego EM, Persoons L, Daelemans D, Camarasa MJ, Insuasty B, Pérez-Pérez MJ. Cuartas V, et al. Among authors: daelemans d. Molecules. 2019 Nov 21;24(23):4236. doi: 10.3390/molecules24234236. Molecules. 2019. PMID: 31766444 Free PMC article.

5

Iron/Copper Co-Catalyzed Cross-Coupling Reaction for the Synthesis of 6-Substituted 7-Deazapurines and the Corresponding Nucleosides.

Li Q, Persoons L, Daelemans D, Herdewijn P. Li Q, et al. Among authors: daelemans d. J Org Chem. 2020 Jan 17;85(2):403-418. doi: 10.1021/acs.joc.9b02414. Epub 2019 Dec 20. J Org Chem. 2020. PMID: 31858795

6

Drug repurposing: phosphate prodrugs of anticancer and antiviral FDA-approved nucleosides as novel antimicrobials.

Pertusati F, Pileggi E, Richards J, Wootton M, Van Leemputte T, Persoons L, De Coster D, Villanueva X, Daelemans D, Steenackers H, McGuigan C, Serpi M. Pertusati F, et al. Among authors: daelemans d. J Antimicrob Chemother. 2020 Oct 1;75(10):2864-2878. doi: 10.1093/jac/dkaa268. J Antimicrob Chemother. 2020. PMID: 32688391

7

Synthesis of Novel Nitroxoline Analogs with Potent Cathepsin B Exopeptidase Inhibitory Activity.

Van de Walle T, Briand M, Mitrović A, Sosič I, Gobec S, Kos J, Persoons L, Daelemans D, De Jonghe S, Ubiparip Z, Desmet T, Van Hecke K, Mangelinckx S, D'hooghe M. Van de Walle T, et al. Among authors: daelemans d, d hooghe m. ChemMedChem. 2020 Dec 15;15(24):2477-2490. doi: 10.1002/cmdc.202000402. Epub 2020 Sep 21. ChemMedChem. 2020. PMID: 32744405

8

Synthesis and Antitumor Activity of C-7-Alkynylated and Arylated Pyrrolotriazine C-Ribonucleosides.

Li Q, Groaz E, Persoons L, Daelemans D, Herdewijn P. Li Q, et al. Among authors: daelemans d. ACS Med Chem Lett. 2020 Jul 9;11(8):1605-1610. doi: 10.1021/acsmedchemlett.0c00269. eCollection 2020 Aug 13. ACS Med Chem Lett. 2020. PMID: 32832030 Free PMC article.

9

Design, synthesis and biological evaluation of pyrazolo[3,4-d]pyrimidine-based protein kinase D inhibitors.

Gilles P, Kashyap RS, Freitas MJ, Ceusters S, Van Asch K, Janssens A, De Jonghe S, Persoons L, Cobbaut M, Daelemans D, Van Lint J, Voet ARD, De Borggraeve WM. Gilles P, et al. Among authors: daelemans d. Eur J Med Chem. 2020 Nov 1;205:112638. doi: 10.1016/j.ejmech.2020.112638. Epub 2020 Jul 29. Eur J Med Chem. 2020. PMID: 32835918

10

N-substituted benzimidazole acrylonitriles as in vitro tubulin polymerization inhibitors: Synthesis, biological activity and computational analysis.

Perin N, Hok L, Beč A, Persoons L, Vanstreels E, Daelemans D, Vianello R, Hranjec M. Perin N, et al. Among authors: daelemans d. Eur J Med Chem. 2021 Feb 5;211:113003. doi: 10.1016/j.ejmech.2020.113003. Epub 2020 Nov 7. Eur J Med Chem. 2021. PMID: 33248847

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