Tomita K - Search Results

1

Discovery of tricyclic HIV-1 integrase-LEDGF/p75 allosteric inhibitors by intramolecular direct arylation reaction.

Taoda Y, Akiyama T, Tomita K, Fujiwara-Kitamura M, Tamura Y, Kawasuji T, Matsuoka E, Akihisa E, Seki T, Yoshinaga T. Taoda Y, et al. Among authors: tomita k. Bioorg Med Chem Lett. 2022 May 15;64:128664. doi: 10.1016/j.bmcl.2022.128664. Epub 2022 Mar 8. Bioorg Med Chem Lett. 2022. PMID: 35272008

2

Discovery of novel 5-hydroxy-4-pyridone-3-carboxy acids as potent inhibitors of influenza Cap-dependent endonuclease.

Miyagawa M, Akiyama T, Mikamiyama-Iwata M, Hattori K, Kurihara N, Taoda Y, Takahashi-Kageyama C, Kurose N, Mikamiyama H, Suzuki N, Takaya K, Tomita K, Matsuo K, Morimoto K, Yoshida R, Shishido T, Yoshinaga T, Sato A, Kawai M. Miyagawa M, et al. Among authors: tomita k. Bioorg Med Chem Lett. 2016 Oct 1;26(19):4739-4742. doi: 10.1016/j.bmcl.2016.08.038. Epub 2016 Aug 18. Bioorg Med Chem Lett. 2016. PMID: 27568084

3

Discovery of novel integrase-LEDGF/p75 allosteric inhibitors based on a benzene scaffold.

Sugiyama S, Iwaki T, Tamura Y, Tomita K, Matsuoka E, Arita S, Seki T, Yoshinaga T, Kawasuji T. Sugiyama S, et al. Among authors: tomita k. Bioorg Med Chem. 2020 Sep 1;28(17):115643. doi: 10.1016/j.bmc.2020.115643. Epub 2020 Jul 10. Bioorg Med Chem. 2020. PMID: 32773094

4

Dihydrodibenzothiepine: Promising hydrophobic pharmacophore in the influenza cap-dependent endonuclease inhibitor.

Taoda Y, Miyagawa M, Akiyama T, Tomita K, Hasegawa Y, Yoshida R, Noshi T, Shishido T, Kawai M. Taoda Y, et al. Among authors: tomita k. Bioorg Med Chem Lett. 2020 Nov 15;30(22):127547. doi: 10.1016/j.bmcl.2020.127547. Epub 2020 Sep 11. Bioorg Med Chem Lett. 2020. PMID: 32927030

5

Synthesis and SAR Study of Carbamoyl Pyridone Bicycle Derivatives as Potent Inhibitors of Influenza Cap-dependent Endonuclease.

Miyagawa M, Akiyama T, Taoda Y, Takaya K, Takahashi-Kageyama C, Tomita K, Yasuo K, Hattori K, Shano S, Yoshida R, Shishido T, Yoshinaga T, Sato A, Kawai M. Miyagawa M, et al. Among authors: tomita k. J Med Chem. 2019 Sep 12;62(17):8101-8114. doi: 10.1021/acs.jmedchem.9b00861. Epub 2019 Aug 19. J Med Chem. 2019. PMID: 31386363

6

Structure-activity relationship study on small peptidic GPR54 agonists.

Tomita K, Niida A, Oishi S, Ohno H, Cluzeau J, Navenot JM, Wang ZX, Peiper SC, Fujii N. Tomita K, et al. Bioorg Med Chem. 2006 Nov 15;14(22):7595-603. doi: 10.1016/j.bmc.2006.07.009. Epub 2006 Aug 1. Bioorg Med Chem. 2006. PMID: 16879969

7

Design and synthesis of downsized metastin (45-54) analogs with maintenance of high GPR54 agonistic activity.

Niida A, Wang Z, Tomita K, Oishi S, Tamamura H, Otaka A, Navenot JM, Broach JR, Peiper SC, Fujii N. Niida A, et al. Among authors: tomita k. Bioorg Med Chem Lett. 2006 Jan 1;16(1):134-7. doi: 10.1016/j.bmcl.2005.09.054. Epub 2005 Oct 18. Bioorg Med Chem Lett. 2006. PMID: 16242330

8

Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres.

Kobayashi K, Oishi S, Hayashi R, Tomita K, Kubo T, Tanahara N, Ohno H, Yoshikawa Y, Furuya T, Hoshino M, Fujii N. Kobayashi K, et al. Among authors: tomita k. J Med Chem. 2012 Mar 22;55(6):2746-57. doi: 10.1021/jm2016914. Epub 2012 Mar 6. J Med Chem. 2012. PMID: 22352868

9

Structure-activity relationship study on polyglutamine binding peptide QBP1.

Tomita K, Popiel HA, Nagai Y, Toda T, Yoshimitsu Y, Ohno H, Oishi S, Fujii N. Tomita K, et al. Bioorg Med Chem. 2009 Feb 1;17(3):1259-63. doi: 10.1016/j.bmc.2008.12.018. Epub 2008 Dec 24. Bioorg Med Chem. 2009. PMID: 19121945

10

Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase.

Tomita K, Oishi S, Ohno H, Peiper SC, Fujii N. Tomita K, et al. J Med Chem. 2008 Dec 11;51(23):7645-9. doi: 10.1021/jm800930w. J Med Chem. 2008. PMID: 19007202

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