Schirmeister T - Search Results

1

Selective noncovalent proteasome inhibiting activity of trifluoromethyl-containing gem-quaternary aziridines.

Ielo L, Patamia V, Citarella A, Schirmeister T, Stagno C, Rescifina A, Micale N, Pace V. Ielo L, et al. Among authors: schirmeister t. Arch Pharm (Weinheim). 2023 Jul;356(7):e2300174. doi: 10.1002/ardp.202300174. Epub 2023 Apr 29. Arch Pharm (Weinheim). 2023. PMID: 37119396 Free article.

2

Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines.

Ielo L, Patamia V, Citarella A, Efferth T, Shahhamzehei N, Schirmeister T, Stagno C, Langer T, Rescifina A, Micale N, Pace V. Ielo L, et al. Among authors: schirmeister t. Int J Mol Sci. 2022 Oct 15;23(20):12363. doi: 10.3390/ijms232012363. Int J Mol Sci. 2022. PMID: 36293216 Free PMC article.

3

Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 M^pro.

Citarella A, Moi D, Pedrini M, Pérez-Peña H, Pieraccini S, Stagno C, Micale N, Schirmeister T, Sibille G, Gribaudo G, Silvani A, Passarella D, Giannini C. Citarella A, et al. Among authors: schirmeister t. Molecules. 2023 Jan 4;28(2):514. doi: 10.3390/molecules28020514. Molecules. 2023. PMID: 36677572 Free PMC article.

4

Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 M^pro Inhibitors.

Fassi EMA, Manenti M, Citarella A, Dei Cas M, Casati S, Micale N, Schirmeister T, Roda G, Silvani A, Grazioso G. Fassi EMA, et al. Among authors: schirmeister t. Molecules. 2023 Mar 3;28(5):2356. doi: 10.3390/molecules28052356. Molecules. 2023. PMID: 36903597 Free PMC article.

5

Synthesis of SARS-CoV-2 M^pro inhibitors bearing a cinnamic ester warhead with in vitro activity against human coronaviruses.

Citarella A, Moi D, Pedrini M, Pérez-Peña H, Pieraccini S, Dimasi A, Stagno C, Micale N, Schirmeister T, Sibille G, Gribaudo G, Silvani A, Giannini C, Passarella D. Citarella A, et al. Among authors: schirmeister t. Org Biomol Chem. 2023 May 10;21(18):3811-3824. doi: 10.1039/d3ob00381g. Org Biomol Chem. 2023. PMID: 37078164 Free article.

6

Two palladium (II) complexes derived from halogen-substituted Schiff bases and 2-picolylamine induce parthanatos-type cell death in sensitive and multi-drug resistant CCRF-CEM leukemia cells.

Zhou M, Boulos JC, Omer EA, Rudbari HA, Schirmeister T, Micale N, Efferth T. Zhou M, et al. Among authors: schirmeister t. Eur J Pharmacol. 2023 Oct 5;956:175980. doi: 10.1016/j.ejphar.2023.175980. Epub 2023 Aug 9. Eur J Pharmacol. 2023. PMID: 37567459

7

Investigating the Cytotoxicity of Ru(II) Polypyridyl Complexes by Changing the Electronic Structure of Salicylaldehyde Ligands.

Taghizadeh Shool M, Amiri Rudbari H, Cuevas-Vicario JV, Rodríguez-Rubio A, Stagno C, Iraci N, Efferth T, Omer EA, Schirmeister T, Blacque O, Moini N, Sheibani E, Micale N. Taghizadeh Shool M, et al. Among authors: schirmeister t. Inorg Chem. 2024 Jan 15;63(2):1083-1101. doi: 10.1021/acs.inorgchem.3c03414. Epub 2023 Dec 29. Inorg Chem. 2024. PMID: 38156413 Free PMC article.

8

Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells.

Citarella A, Petrella S, Moi D, Dimasi A, Braga T, Ruberto L, Pieraccini S, Sironi M, Micale N, Schirmeister T, Damia G, Fasano V, Silvani A, Giannini C, Passarella D. Citarella A, et al. Among authors: schirmeister t. Bioorg Med Chem. 2024 Dec 1;115:117987. doi: 10.1016/j.bmc.2024.117987. Epub 2024 Nov 5. Bioorg Med Chem. 2024. PMID: 39509759

9

Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria.

Di Chio C, Starvaggi J, Totaro N, Previti S, Natale B, Cosconati S, Bogacz M, Schirmeister T, Legac J, Rosenthal PJ, Zappalà M, Ettari R. Di Chio C, et al. Among authors: schirmeister t. Int J Mol Sci. 2024 Apr 17;25(8):4410. doi: 10.3390/ijms25084410. Int J Mol Sci. 2024. PMID: 38673995 Free PMC article.

10

Covalent S-Adenosylhomocysteine-Based DNA Methyltransferase 2 Inhibitors with a New Type of Aryl Warhead.

Schwickert M, Zimmermann RA, Habeck T, Hoba SN, Nidoieva Z, Fischer TR, Stark MM, Kersten C, Lermyte F, Helm M, Schirmeister T. Schwickert M, et al. Among authors: schirmeister t. ACS Med Chem Lett. 2023 May 9;14(6):777-787. doi: 10.1021/acsmedchemlett.3c00062. eCollection 2023 Jun 8. ACS Med Chem Lett. 2023. PMID: 37312859 Free PMC article.

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