Discovery and Functional Characterization of a Potent, Selective, and Metabolically Stable PROTAC of the Protein Kinases DYRK1A and DYRK1B.
Wilms G, Schofield K, Maddern S, Foley C, Shaw Y, Smith B, Basantes LE, Schwandt K, Babendreyer A, Chavez T, McKee N, Gokhale V, Kallabis S, Meissner F, Rokey SN, Dunckley T, Montfort WR, Becker W, Hulme C.
Wilms G, et al. Among authors: schofield k.
J Med Chem. 2024 Oct 10;67(19):17259-17289. doi: 10.1021/acs.jmedchem.4c01130. Epub 2024 Sep 30.
J Med Chem. 2024.
PMID: 39344427