Jacobson KA - Search Results

1

Structural Modification and Biological Evaluation of 2,8-Disubstituted Adenine and Its Nucleosides as A_2A Adenosine Receptor Antagonists: Exploring the Roles of Ribose at Adenosine Receptors.

Kim G, Jarhad DB, Lee G, Kim G, Hou X, Yu J, Lee CS, Warnick E, Gao ZG, Ahn SY, Kwak D, Park K, Lee SD, Park TU, Jung SY, Lee JH, Choi JR, Kim M, Kim D, Kim B, Jacobson KA, Jeong LS. Kim G, et al. Among authors: jacobson ka. J Med Chem. 2024 Jun 27;67(12):10490-10507. doi: 10.1021/acs.jmedchem.4c01003. Epub 2024 Jun 6. J Med Chem. 2024. PMID: 38845345

2

Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists.

Jacobson KA, Nikodijevic O, Ji XD, Berkich DA, Eveleth D, Dean RL, Hiramatsu K, Kassell NF, van Galen PJ, Lee KS, et al. Jacobson KA, et al. J Med Chem. 1992 Oct 30;35(22):4143-9. doi: 10.1021/jm00100a020. J Med Chem. 1992. PMID: 1433217 Free PMC article.

3

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.

Jacobson KA, van Galen PJ, Williams M. Jacobson KA, et al. J Med Chem. 1992 Feb 7;35(3):407-22. doi: 10.1021/jm00081a001. J Med Chem. 1992. PMID: 1738138 Free PMC article. Review. No abstract available.

4

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.

Jacobson KA, Barone S, Kammula U, Stiles GL. Jacobson KA, et al. J Med Chem. 1989 May;32(5):1043-51. doi: 10.1021/jm00125a019. J Med Chem. 1989. PMID: 2709373 Free PMC article.

5

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

Jacobson KA, Kiriasis L, Barone S, Bradbury BJ, Kammula U, Campagne JM, Secunda S, Daly JW, Neumeyer JL, Pfleiderer W. Jacobson KA, et al. J Med Chem. 1989 Aug;32(8):1873-9. doi: 10.1021/jm00128a031. J Med Chem. 1989. PMID: 2754711 Free PMC article.

6

Search for new purine- and ribose-modified adenosine analogues as selective agonists and antagonists at adenosine receptors.

Siddiqi SM, Jacobson KA, Esker JL, Olah ME, Ji XD, Melman N, Tiwari KN, Secrist JA 3rd, Schneller SW, Cristalli G, et al. Siddiqi SM, et al. Among authors: jacobson ka. J Med Chem. 1995 Mar 31;38(7):1174-88. doi: 10.1021/jm00007a014. J Med Chem. 1995. PMID: 7707320 Free PMC article.

7

Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors.

Jacobson KA, Siddiqi SM, Olah ME, Ji XD, Melman N, Bellamkonda K, Meshulam Y, Stiles GL, Kim HO. Jacobson KA, et al. J Med Chem. 1995 May 12;38(10):1720-35. doi: 10.1021/jm00010a017. J Med Chem. 1995. PMID: 7752196 Free PMC article.

8

Structure-activity relationships of 1,3-dialkylxanthine derivatives at rat A3 adenosine receptors.

Kim HO, Ji XD, Melman N, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Sep 30;37(20):3373-82. doi: 10.1021/jm00046a022. J Med Chem. 1994. PMID: 7932565 Free PMC article.

9

2-Substitution of N6-benzyladenosine-5'-uronamides enhances selectivity for A3 adenosine receptors.

Kim HO, Ji XD, Siddiqi SM, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Oct 14;37(21):3614-21. doi: 10.1021/jm00047a018. J Med Chem. 1994. PMID: 7932588 Free PMC article.

10

Selective ligands for rat A3 adenosine receptors: structure-activity relationships of 1,3-dialkylxanthine 7-riboside derivatives.

Kim HO, Ji XD, Melman N, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Nov 11;37(23):4020-30. doi: 10.1021/jm00049a021. J Med Chem. 1994. PMID: 7966162 Free PMC article.

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