Metzger E - Search Results

1

Structure-Activity Studies of 1,2,4-Oxadiazoles for the Inhibition of the NAD⁺-Dependent Lysine Deacylase Sirtuin 2.

Colcerasa A, Friedrich F, Melesina J, Moser P, Vogelmann A, Tzortzoglou P, Neuwirt E, Sum M, Robaa D, Zhang L, Ramos-Morales E, Romier C, Einsle O, Metzger E, Schüle R, Groß O, Sippl W, Jung M. Colcerasa A, et al. Among authors: metzger e. J Med Chem. 2024 Jun 27;67(12):10076-10095. doi: 10.1021/acs.jmedchem.4c00229. Epub 2024 Jun 7. J Med Chem. 2024. PMID: 38847803

2

A novel inducible transactivation domain in the androgen receptor: implications for PRK in prostate cancer.

Metzger E, Müller JM, Ferrari S, Buettner R, Schüle R. Metzger E, et al. EMBO J. 2003 Jan 15;22(2):270-80. doi: 10.1093/emboj/cdg023. EMBO J. 2003. PMID: 12514133 Free PMC article.

3

Histone demethylation and androgen-dependent transcription.

Metzger E, Wissmann M, Schüle R. Metzger E, et al. Curr Opin Genet Dev. 2006 Oct;16(5):513-7. doi: 10.1016/j.gde.2006.08.013. Epub 2006 Aug 17. Curr Opin Genet Dev. 2006. PMID: 16919442 Review.

4

The expanding world of histone lysine demethylases.

Metzger E, Schüle R. Metzger E, et al. Nat Struct Mol Biol. 2007 Apr;14(4):252-4. doi: 10.1038/nsmb0407-252. Nat Struct Mol Biol. 2007. PMID: 17410086 No abstract available.

5

Target-based approach to inhibitors of histone arginine methyltransferases.

Spannhoff A, Heinke R, Bauer I, Trojer P, Metzger E, Gust R, Schüle R, Brosch G, Sippl W, Jung M. Spannhoff A, et al. Among authors: metzger e. J Med Chem. 2007 May 17;50(10):2319-25. doi: 10.1021/jm061250e. Epub 2007 Apr 14. J Med Chem. 2007. PMID: 17432842

6

Acyl derivatives of p-aminosulfonamides and dapsone as new inhibitors of the arginine methyltransferase hPRMT1.

Bissinger EM, Heinke R, Spannhoff A, Eberlin A, Metzger E, Cura V, Hassenboehler P, Cavarelli J, Schüle R, Bedford MT, Sippl W, Jung M. Bissinger EM, et al. Among authors: metzger e. Bioorg Med Chem. 2011 Jun 15;19(12):3717-31. doi: 10.1016/j.bmc.2011.02.032. Epub 2011 Feb 27. Bioorg Med Chem. 2011. PMID: 21440447

7

Screening assays for epigenetic targets using native histones as substrates.

Hauser AT, Bissinger EM, Metzger E, Repenning A, Bauer UM, Mai A, Schüle R, Jung M. Hauser AT, et al. Among authors: metzger e. J Biomol Screen. 2012 Jan;17(1):18-26. doi: 10.1177/1087057111423968. Epub 2011 Sep 30. J Biomol Screen. 2012. PMID: 21965113

8

Impairment of prostate cancer cell growth by a selective and reversible lysine-specific demethylase 1 inhibitor.

Willmann D, Lim S, Wetzel S, Metzger E, Jandausch A, Wilk W, Jung M, Forne I, Imhof A, Janzer A, Kirfel J, Waldmann H, Schüle R, Buettner R. Willmann D, et al. Among authors: metzger e. Int J Cancer. 2012 Dec 1;131(11):2704-9. doi: 10.1002/ijc.27555. Epub 2012 Jun 28. Int J Cancer. 2012. PMID: 22447389

9

Lestaurtinib inhibits histone phosphorylation and androgen-dependent gene expression in prostate cancer cells.

Köhler J, Erlenkamp G, Eberlin A, Rumpf T, Slynko I, Metzger E, Schüle R, Sippl W, Jung M. Köhler J, et al. Among authors: metzger e. PLoS One. 2012;7(4):e34973. doi: 10.1371/journal.pone.0034973. Epub 2012 Apr 20. PLoS One. 2012. PMID: 22532837 Free PMC article.

10

Nonpeptidic propargylamines as inhibitors of lysine specific demethylase 1 (LSD1) with cellular activity.

Schmitt ML, Hauser AT, Carlino L, Pippel M, Schulz-Fincke J, Metzger E, Willmann D, Yiu T, Barton M, Schüle R, Sippl W, Jung M. Schmitt ML, et al. Among authors: metzger e. J Med Chem. 2013 Sep 26;56(18):7334-42. doi: 10.1021/jm400792m. Epub 2013 Sep 5. J Med Chem. 2013. PMID: 24007511 Free PMC article.

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