Salmaso V - Search Results

1

7-Amino-[1,2,4]triazolo[1,5-a][1,3,5]triazines as CK1δ inhibitors: Exploring substitutions at the 2 and 5-positions.

Grieco I, Bassani D, Trevisan L, Salmaso V, Cescon E, Prencipe F, Da Ros T, Martinez-Gonzalez L, Martinez A, Spalluto G, Moro S, Federico S. Grieco I, et al. Among authors: salmaso v. Bioorg Chem. 2024 Oct;151:107659. doi: 10.1016/j.bioorg.2024.107659. Epub 2024 Jul 17. Bioorg Chem. 2024. PMID: 39059072 Free article.

2

Lipid Trolling to Optimize A₃ Adenosine Receptor-Positive Allosteric Modulators (PAMs).

Pradhan B, Pavan M, Fisher CL, Salmaso V, Wan TC, Keyes RF, Rollison N, Suresh RR, Kumar TS, Gao ZG, Smith BC, Auchampach JA, Jacobson KA. Pradhan B, et al. Among authors: salmaso v. J Med Chem. 2024 Jul 25;67(14):12221-12247. doi: 10.1021/acs.jmedchem.4c00944. Epub 2024 Jul 3. J Med Chem. 2024. PMID: 38959401

3

Structural Investigations on 2-Amidobenzimidazole Derivatives as New Inhibitors of Protein Kinase CK1 Delta.

Calenda S, Catarzi D, Varano F, Vigiani E, Volpini R, Lambertucci C, Spinaci A, Trevisan L, Grieco I, Federico S, Spalluto G, Novello G, Salmaso V, Moro S, Colotta V. Calenda S, et al. Among authors: salmaso v. Pharmaceuticals (Basel). 2024 Apr 7;17(4):468. doi: 10.3390/ph17040468. Pharmaceuticals (Basel). 2024. PMID: 38675428 Free PMC article.

4

Extrahelical Binding Site for a 1H-Imidazo[4,5-c]quinolin-4-amine A₃ Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7.

Fisher CL, Pavan M, Salmaso V, Keyes RF, Wan TC, Pradhan B, Gao ZG, Smith BC, Jacobson KA, Auchampach JA. Fisher CL, et al. Among authors: salmaso v. Mol Pharmacol. 2024 Feb 15;105(3):213-223. doi: 10.1124/molpharm.123.000784. Mol Pharmacol. 2024. PMID: 38182432 Free PMC article.

5

2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A₁ Adenosine Receptor Positive Allosteric Modulators.

Oliva P, Suresh RR, Pasquini S, Salmaso V, Will EJ, Tosh DK, Gao ZG, Liu N, Gavrilova O, Vincenzi F, Varani K, Jacobson KA. Oliva P, et al. Among authors: salmaso v. ACS Med Chem Lett. 2023 Nov 13;14(12):1640-1646. doi: 10.1021/acsmedchemlett.3c00315. eCollection 2023 Dec 14. ACS Med Chem Lett. 2023. PMID: 38116442

6

Thermal titration molecular dynamics (TTMD): shedding light on the stability of RNA-small molecule complexes.

Dodaro A, Pavan M, Menin S, Salmaso V, Sturlese M, Moro S. Dodaro A, et al. Among authors: salmaso v. Front Mol Biosci. 2023 Nov 13;10:1294543. doi: 10.3389/fmolb.2023.1294543. eCollection 2023. Front Mol Biosci. 2023. PMID: 38028536 Free PMC article.

7

Pyrazolo-triazolo-pyrimidine Scaffold as a Molecular Passepartout for the Pan-Recognition of Human Adenosine Receptors.

Salmaso V, Persico M, Da Ros T, Spalluto G, Kachler S, Klotz KN, Moro S, Federico S. Salmaso V, et al. Biomolecules. 2023 Nov 3;13(11):1610. doi: 10.3390/biom13111610. Biomolecules. 2023. PMID: 38002292 Free PMC article.

8

Stereocontrolled access to thioisosteres of nucleoside di- and triphosphates.

Zhang HJ, Ociepa M, Nassir M, Zheng B, Lewicki SA, Salmaso V, Baburi H, Nagel J, Mirza S, Bueschbell B, Al-Hroub H, Perzanowska O, Lin Z, Schmidt MA, Eastgate MD, Jacobson KA, Müller CE, Kowalska J, Jemielity J, Baran PS. Zhang HJ, et al. Among authors: salmaso v. Nat Chem. 2024 Feb;16(2):249-258. doi: 10.1038/s41557-023-01347-2. Epub 2023 Oct 19. Nat Chem. 2024. PMID: 37857844

9

First Potent Macrocyclic A₃ Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences.

Tosh DK, Fisher CL, Salmaso V, Wan TC, Campbell RG, Chen E, Gao ZG, Auchampach JA, Jacobson KA. Tosh DK, et al. Among authors: salmaso v. ACS Pharmacol Transl Sci. 2023 Aug 8;6(9):1288-1305. doi: 10.1021/acsptsci.3c00126. eCollection 2023 Sep 8. ACS Pharmacol Transl Sci. 2023. PMID: 37705595 Free PMC article.

10

[1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A₃ Adenosine Receptors in Cancer Cell Lines.

Federico S, Persico M, Trevisan L, Biasinutto C, Bolcato G, Salmaso V, Da Ros T, Gianferrara T, Prencipe F, Kachler S, Klotz KN, Pacor S, Moro S, Spalluto G. Federico S, et al. Among authors: salmaso v. ChemMedChem. 2023 Nov 2;18(21):e202300299. doi: 10.1002/cmdc.202300299. Epub 2023 Sep 22. ChemMedChem. 2023. PMID: 37675643

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