Leurs R - Search Results

1

Conformational dynamics underlying atypical chemokine receptor 3 activation.

Otun O, Aljamous C, Del Nero E, Arimont-Segura M, Bosma R, Zarzycka B, Girbau T, Leyrat C, de Graaf C, Leurs R, Durroux T, Granier S, Cong X, Bechara C. Otun O, et al. Among authors: leurs r. Proc Natl Acad Sci U S A. 2024 Jul 23;121(30):e2404000121. doi: 10.1073/pnas.2404000121. Epub 2024 Jul 15. Proc Natl Acad Sci U S A. 2024. PMID: 39008676 Free PMC article.

2

Predicting the target landscape of kinase inhibitors using 3D convolutional neural networks.

Kanev GK, Zhang Y, Kooistra AJ, Bender A, Leurs R, Bailey D, Würdinger T, de Graaf C, de Esch IJP, Westerman BA. Kanev GK, et al. Among authors: leurs r. PLoS Comput Biol. 2023 Sep 5;19(9):e1011301. doi: 10.1371/journal.pcbi.1011301. eCollection 2023 Sep. PLoS Comput Biol. 2023. PMID: 37669273 Free PMC article.

3

Ligand-directed biased agonism at human histamine H₃ receptor isoforms across Gα_i/o- and β-arrestin2-mediated pathways.

Rahman SN, Imhaouran F, Leurs R, Christopoulos A, Valant C, Langmead CJ. Rahman SN, et al. Among authors: leurs r. Biochem Pharmacol. 2024 Oct;228:115988. doi: 10.1016/j.bcp.2023.115988. Epub 2023 Dec 28. Biochem Pharmacol. 2024. PMID: 38159685 Free article.

4

Aquaporin-4 and GPRC5B: old and new players in controlling brain oedema.

Passchier EMJ, Kerst S, Brouwers E, Hamilton EMC, Bisseling Q, Bugiani M, Waisfisz Q, Kitchen P, Unger L, Breur M, Hoogterp L, de Vries SI, Abbink TEM, Kole MHP, Leurs R, Vischer HF, Brignone MS, Ambrosini E, Feillet F, Born AP, Epstein LG, Mansvelder HD, Min R, van der Knaap MS. Passchier EMJ, et al. Among authors: leurs r. Brain. 2023 Aug 1;146(8):3444-3454. doi: 10.1093/brain/awad146. Brain. 2023. PMID: 37143309 Free PMC article.

5

The Role of Water Networks in Phosphodiesterase Inhibitor Dissociation and Kinetic Selectivity.

Blaazer AR, Singh AK, Zara L, Boronat P, Bautista LJ, Irving S, Majewski M, Barril X, Wijtmans M, Danielson UH, Sterk GJ, Leurs R, van Muijlwijk-Koezen JE, Brown DG, de Esch IJP. Blaazer AR, et al. Among authors: leurs r. ChemMedChem. 2024 Nov 18;19(22):e202400417. doi: 10.1002/cmdc.202400417. Epub 2024 Sep 12. ChemMedChem. 2024. PMID: 39193819

6

Adhesion of Crithidia fasciculata promotes a rapid change in developmental fate driven by cAMP signaling.

Denecke S, Malfara MF, Hodges KR, Holmes NA, Williams AR, Gallagher-Teske JH, Pascarella JM, Daniels AM, Sterk GJ, Leurs R, Ruthel G, Hoang R, Povelones ML, Povelones M. Denecke S, et al. Among authors: leurs r. mSphere. 2024 Oct 29;9(10):e0061724. doi: 10.1128/msphere.00617-24. Epub 2024 Sep 24. mSphere. 2024. PMID: 39315810 Free PMC article.

7

Pharmacological characterization of the zebrafish Hrh2a histamine H₂ receptor.

McNaught-Flores DA, Chen YC, Arias-Montaño JA, Panula P, Leurs R. McNaught-Flores DA, et al. Among authors: leurs r. Eur J Pharmacol. 2024 Oct 15;981:176870. doi: 10.1016/j.ejphar.2024.176870. Epub 2024 Aug 6. Eur J Pharmacol. 2024. PMID: 39117262 Free article.

8

Histamine H₃ Receptor Isoforms: Insights from Alternative Splicing to Functional Complexity.

Gao M, Ooms JF, Leurs R, Vischer HF. Gao M, et al. Among authors: leurs r. Biomolecules. 2024 Jun 26;14(7):761. doi: 10.3390/biom14070761. Biomolecules. 2024. PMID: 39062475 Free PMC article. Review.

9

A high-affinity, cis-on photoswitchable beta blocker to optically control β₂-adrenergic receptors in vitro and in vivo.

Shi S, Zheng Y, Goulding J, Marri S, Lucarini L, Konecny B, Sgambellone S, Villano S, Bosma R, Wijtmans M, Briddon SJ, Zarzycka BA, Vischer HF, Leurs R. Shi S, et al. Among authors: leurs r. Biochem Pharmacol. 2024 Aug;226:116396. doi: 10.1016/j.bcp.2024.116396. Epub 2024 Jun 26. Biochem Pharmacol. 2024. PMID: 38942089 Free article.

10

Multiplex Detection of Fluorescent Chemokine Binding to CXC Chemokine Receptors by NanoBRET.

Adamska JM, Leftheriotis S, Bosma R, Vischer HF, Leurs R. Adamska JM, et al. Among authors: leurs r. Int J Mol Sci. 2024 May 4;25(9):5018. doi: 10.3390/ijms25095018. Int J Mol Sci. 2024. PMID: 38732237 Free PMC article.

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