Tasso B - Search Results

1

Discovery of Novel Thiazole-Based SIRT2 Inhibitors as Anticancer Agents: Molecular Modeling, Chemical Synthesis and Biological Assays.

Piacente F, Guccione G, Scarano N, Lunaccio D, Miro C, Abbotto E, Salis A, Tasso B, Dentice M, Bruzzone S, Cichero E, Millo E. Piacente F, et al. Among authors: tasso b. Int J Mol Sci. 2024 Oct 15;25(20):11084. doi: 10.3390/ijms252011084. Int J Mol Sci. 2024. PMID: 39456864 Free PMC article.

2

Discovery of novel VX-809 hybrid derivatives as F508del-CFTR correctors by molecular modeling, chemical synthesis and biological assays.

Parodi A, Righetti G, Pesce E, Salis A, Tasso B, Urbinati C, Tomati V, Damonte G, Rusnati M, Pedemonte N, Cichero E, Millo E. Parodi A, et al. Among authors: tasso b. Eur J Med Chem. 2020 Dec 15;208:112833. doi: 10.1016/j.ejmech.2020.112833. Epub 2020 Sep 12. Eur J Med Chem. 2020. PMID: 32971410

3

Molecular Docking and QSAR Studies as Computational Tools Exploring the Rescue Ability of F508del CFTR Correctors.

Righetti G, Casale M, Liessi N, Tasso B, Salis A, Tonelli M, Millo E, Pedemonte N, Fossa P, Cichero E. Righetti G, et al. Among authors: tasso b. Int J Mol Sci. 2020 Oct 29;21(21):8084. doi: 10.3390/ijms21218084. Int J Mol Sci. 2020. PMID: 33138251 Free PMC article.

4

Synthesis and biological evaluation of novel thiazole- VX-809 hybrid derivatives as F508del correctors by QSAR-based filtering tools.

Liessi N, Cichero E, Pesce E, Arkel M, Salis A, Tomati V, Paccagnella M, Damonte G, Tasso B, Galietta LJV, Pedemonte N, Fossa P, Millo E. Liessi N, et al. Among authors: tasso b. Eur J Med Chem. 2018 Jan 20;144:179-200. doi: 10.1016/j.ejmech.2017.12.030. Epub 2017 Dec 8. Eur J Med Chem. 2018. PMID: 29272749

5

Differential modulation of SIRT6 deacetylase and deacylase activities by lysine-based small molecules.

Sociali G, Liessi N, Grozio A, Caffa I, Parenti MD, Ravera S, Tasso B, Benzi A, Nencioni A, Del Rio A, Robina I, Millo E, Bruzzone S. Sociali G, et al. Among authors: tasso b. Mol Divers. 2020 Aug;24(3):655-671. doi: 10.1007/s11030-019-09971-2. Epub 2019 Jun 25. Mol Divers. 2020. PMID: 31240519

6

Synthesis and Structure-activity Relationship of Aminoarylthiazole Derivatives as Potential Potentiators of the Chloride Transport Defect in Cystic Fibrosis.

Liessi N, Pesce E, Salis A, Damonte G, Tasso B, Cichero E, Pedemonte N, Millo E. Liessi N, et al. Among authors: tasso b. Med Chem. 2021;17(6):646-657. doi: 10.2174/1573406416666200306114300. Med Chem. 2021. PMID: 32141420

7

Journey on VX-809-Based Hybrid Derivatives towards Drug-like F508del-CFTR Correctors: From Molecular Modeling to Chemical Synthesis and Biological Assays.

Parodi A, Righetti G, Pesce E, Salis A, Tomati V, Pastorino C, Tasso B, Benvenuti M, Damonte G, Pedemonte N, Cichero E, Millo E. Parodi A, et al. Among authors: tasso b. Pharmaceuticals (Basel). 2022 Feb 23;15(3):274. doi: 10.3390/ph15030274. Pharmaceuticals (Basel). 2022. PMID: 35337072 Free PMC article.

8

Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles.

Cichero E, Tonelli M, Novelli F, Tasso B, Delogu I, Loddo R, Bruno O, Fossa P. Cichero E, et al. Among authors: tasso b. J Enzyme Inhib Med Chem. 2017 Dec;32(1):375-402. doi: 10.1080/14756366.2016.1256881. J Enzyme Inhib Med Chem. 2017. PMID: 28276287 Free PMC article.

9

Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction.

Tonelli M, Cichero E, Mahmoud AM, Rabbito A, Tasso B, Fossa P, Ligresti A. Tonelli M, et al. Among authors: tasso b. Medchemcomm. 2018 Oct 10;9(12):2045-2054. doi: 10.1039/c8md00461g. eCollection 2018 Dec 1. Medchemcomm. 2018. PMID: 30647880 Free PMC article.

10

Nanotechnology of Tyrosine Kinase Inhibitors in Cancer Therapy: A Perspective.

Russo E, Spallarossa A, Tasso B, Villa C, Brullo C. Russo E, et al. Among authors: tasso b. Int J Mol Sci. 2021 Jun 18;22(12):6538. doi: 10.3390/ijms22126538. Int J Mol Sci. 2021. PMID: 34207175 Free PMC article. Review.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

62 results

Search Page

Filters