Kassack MU - Search Results

1

Deciphering the Therapeutic Potential of Novel Pentyloxyamide-Based Class I, IIb HDAC Inhibitors against Therapy-Resistant Leukemia.

Fischer F, Schliehe-Diecks J, Tu JW, Gangnus T, Ho YL, Hebeis M, Alves Avelar LA, Scharov K, Watrin T, Kemkes M, Stachura P, Daugs K, Biermann L, Kremeyer J, Horstick N, Span I, Pandyra AA, Borkhardt A, Gohlke H, Kassack MU, Burckhardt BB, Bhatia S, Kurz T. Fischer F, et al. Among authors: kassack mu. J Med Chem. 2024 Nov 27. doi: 10.1021/acs.jmedchem.4c02024. Online ahead of print. J Med Chem. 2024. PMID: 39602240

2

YAK577 Attenuates Cardiac Remodeling and Fibrosis in Isoproterenol-Infused Heart Failure Mice by Downregulating MMP12.

Zhou H, Kee HJ, Wan L, Asfaha Y, Fischer F, Kassack MU, Kurz T, Kim SH, Kee SJ, Hong YJ, Jeong MH. Zhou H, et al. Among authors: kassack mu. Korean Circ J. 2024 Oct 11. doi: 10.4070/kcj.2024.0093. Online ahead of print. Korean Circ J. 2024. PMID: 39601396

3

Multicomponent syntheses enable the discovery of novel quisinostat-derived chemotypes as histone deacetylase inhibitors.

Stopper D, Buntrock S, Tan K, de Carvalho LP, Schäker-Hübner L, Held J, Kassack MU, Hansen FK. Stopper D, et al. Among authors: kassack mu. Eur J Med Chem. 2024 Nov 8;281:117045. doi: 10.1016/j.ejmech.2024.117045. Online ahead of print. Eur J Med Chem. 2024. PMID: 39549507 Free article.

4

Triple Combination of Entinostat, a Bromodomain Inhibitor, and Cisplatin Is a Promising Treatment Option for Bladder Cancer.

Bollmann LM, Lange F, Hamacher A, Biermann L, Schäker-Hübner L, Hansen FK, Kassack MU. Bollmann LM, et al. Among authors: kassack mu. Cancers (Basel). 2024 Oct 2;16(19):3374. doi: 10.3390/cancers16193374. Cancers (Basel). 2024. PMID: 39409994 Free PMC article.

5

Hydrazide-Based Class I Selective HDAC Inhibitors Completely Reverse Chemoresistance Synergistically in Platinum-Resistant Solid Cancer Cells.

Kraft FB, Biermann L, Schäker-Hübner L, Hanl M, Hamacher A, Kassack MU, Hansen FK. Kraft FB, et al. Among authors: kassack mu. J Med Chem. 2024 Oct 10;67(19):17796-17819. doi: 10.1021/acs.jmedchem.4c01817. Epub 2024 Oct 2. J Med Chem. 2024. PMID: 39356226

6

The Antioxidant and HDAC-Inhibitor α-Lipoic Acid Is Synergistic with Exemestane in Estrogen Receptor-Positive Breast Cancer Cells.

Pradel LS, Ho YL, Gohlke H, Kassack MU. Pradel LS, et al. Among authors: kassack mu. Int J Mol Sci. 2024 Aug 2;25(15):8455. doi: 10.3390/ijms25158455. Int J Mol Sci. 2024. PMID: 39126024 Free PMC article.

7

Novel Histone Deacetylase (HDAC) Inhibitor Induces Apoptosis and Suppresses Invasion via E-Cadherin Upregulation in Pancreatic Ductal Adenocarcinoma (PDAC).

Schiedlauske K, Deipenbrock A, Pflieger M, Hamacher A, Hänsel J, Kassack MU, Kurz T, Teusch NE. Schiedlauske K, et al. Among authors: kassack mu. Pharmaceuticals (Basel). 2024 Jun 7;17(6):752. doi: 10.3390/ph17060752. Pharmaceuticals (Basel). 2024. PMID: 38931419 Free PMC article.

8

5-(Trifluoromethyl)-1,2,4-oxadiazole (TFMO)-based highly selective class IIa HDAC inhibitors exhibit synergistic anticancer activity in combination with bortezomib.

Asfaha Y, Bollmann LM, Skerhut AJ, Fischer F, Horstick N, Roth D, Wecker M, Mammen C, Smits SHJ, Fluegen G, Kassack MU, Kurz T. Asfaha Y, et al. Among authors: kassack mu. Eur J Med Chem. 2024 Jan 5;263:115907. doi: 10.1016/j.ejmech.2023.115907. Epub 2023 Nov 10. Eur J Med Chem. 2024. PMID: 37979441

9

Synergistic Interaction of the Class IIa HDAC Inhibitor CHDI0039 with Bortezomib in Head and Neck Cancer Cells.

Schrenk C, Bollmann LM, Haist C, Bister A, Wiek C, Wecker M, Roth D, Petzsch P, Köhrer K, Hamacher A, Hanenberg H, Fluegen G, Kassack MU. Schrenk C, et al. Among authors: kassack mu. Int J Mol Sci. 2023 Mar 14;24(6):5553. doi: 10.3390/ijms24065553. Int J Mol Sci. 2023. PMID: 36982651 Free PMC article.

10

The Novel Class IIa Selective Histone Deacetylase Inhibitor YAK540 Is Synergistic with Bortezomib in Leukemia Cell Lines.

Bollmann LM, Skerhut AJ, Asfaha Y, Horstick N, Hanenberg H, Hamacher A, Kurz T, Kassack MU. Bollmann LM, et al. Among authors: kassack mu. Int J Mol Sci. 2022 Nov 2;23(21):13398. doi: 10.3390/ijms232113398. Int J Mol Sci. 2022. PMID: 36362189 Free PMC article.

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