Merchant KJ - Search Results

1

Identification of L-tryptophan derivatives with potent and selective antagonist activity at the NK1 receptor.

MacLeod AM, Merchant KJ, Brookfield F, Kelleher F, Stevenson G, Owens AP, Swain CJ, Casiceri MA, Sadowski S, Ber E, et al. MacLeod AM, et al. Among authors: merchant kj. J Med Chem. 1994 Apr 29;37(9):1269-74. doi: 10.1021/jm00035a006. J Med Chem. 1994. PMID: 7513763

2

Synthesis and biological activity of 1,2,4-oxadiazole derivatives: highly potent and efficacious agonists for cortical muscarinic receptors.

Street LJ, Baker R, Book T, Kneen CO, MacLeod AM, Merchant KJ, Showell GA, Saunders J, Herbert RH, Freedman SB, et al. Street LJ, et al. Among authors: merchant kj. J Med Chem. 1990 Oct;33(10):2690-7. doi: 10.1021/jm00172a003. J Med Chem. 1990. PMID: 2213823

3

Novel quinuclidine-based ligands for the muscarinic cholinergic receptor.

Saunders J, Cassidy M, Freedman SB, Harley EA, Iversen LL, Kneen C, MacLeod AM, Merchant KJ, Snow RJ, Baker R. Saunders J, et al. Among authors: merchant kj. J Med Chem. 1990 Apr;33(4):1128-38. doi: 10.1021/jm00166a008. J Med Chem. 1990. PMID: 2319559

4

Synthesis and muscarinic activities of 1,2,4-thiadiazoles.

MacLeod AM, Baker R, Freedman SB, Patel S, Merchant KJ, Roe M, Saunders J. MacLeod AM, et al. Among authors: merchant kj. J Med Chem. 1990 Jul;33(7):2052-9. doi: 10.1021/jm00169a041. J Med Chem. 1990. PMID: 2362286

5

Identification of a series of 3-(benzyloxy)-1-azabicyclo[2.2.2]octane human NK1 antagonists.

Swain CJ, Seward EM, Cascieri MA, Fong TM, Herbert R, MacIntyre DE, Merchant KJ, Owen SN, Owens AP, Sabin V, et al. Swain CJ, et al. Among authors: merchant kj. J Med Chem. 1995 Nov 24;38(24):4793-805. doi: 10.1021/jm00024a007. J Med Chem. 1995. PMID: 7490729

6

Characterization of the interaction of N-acyl-L-tryptophan benzyl ester neurokinin antagonists with the human neurokinin-1 receptor.

Cascieri MA, Macleod AM, Underwood D, Shiao LL, Ber E, Sadowski S, Yu H, Merchant KJ, Swain CJ, Strader CD, et al. Cascieri MA, et al. Among authors: merchant kj. J Biol Chem. 1994 Mar 4;269(9):6587-91. J Biol Chem. 1994. PMID: 7509807 Free article.

7

Synthesis and biological evaluation of NK1 antagonists derived from L-tryptophan.

MacLeod AM, Cascieri MA, Merchant KJ, Sadowski S, Hardwicke S, Lewis RT, MacIntyre DE, Metzger JM, Fong TM, Shepheard S, et al. MacLeod AM, et al. Among authors: merchant kj. J Med Chem. 1995 Mar 17;38(6):934-41. doi: 10.1021/jm00006a012. J Med Chem. 1995. PMID: 7535362

8

Tryptophan-derived NK1 antagonists: conformationally constrained heterocyclic bioisosteres of the ester linkage.

Lewis RT, Macleod AM, Merchant KJ, Kelleher F, Sanderson I, Herbert RH, Cascieri MA, Sadowski S, Ball RG, Hoogsteen K. Lewis RT, et al. Among authors: merchant kj. J Med Chem. 1995 Mar 17;38(6):923-33. doi: 10.1021/jm00006a011. J Med Chem. 1995. PMID: 7699709

9

N-acyl-L-tryptophan benzyl esters: potent substance P receptor antagonists.

MacLeod AM, Merchant KJ, Cascieri MA, Sadowski S, Ber E, Swain CJ, Baker R. MacLeod AM, et al. Among authors: merchant kj. J Med Chem. 1993 Jul 9;36(14):2044-5. doi: 10.1021/jm00066a015. J Med Chem. 1993. PMID: 8393115 No abstract available.

10

4,4-Disubstituted piperidine high-affinity NK1 antagonists: structure-activity relationships and in vivo activity.

Stevenson GI, Huscroft I, MacLeod AM, Swain CJ, Cascieri MA, Chicchi GG, Graham MI, Harrison T, Kelleher FJ, Kurtz M, Ladduwahetty T, Merchant KJ, Metzger JM, MacIntyre DE, Sadowski S, Sohal B, Owens AP. Stevenson GI, et al. Among authors: merchant kj. J Med Chem. 1998 Nov 5;41(23):4623-35. doi: 10.1021/jm980376b. J Med Chem. 1998. PMID: 9804702

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