Talley JJ - Search Results

1

Discovery of a novel class of potent HIV-1 protease inhibitors containing the (R)-(hydroxyethyl)urea isostere.

Getman DP, DeCrescenzo GA, Heintz RM, Reed KL, Talley JJ, Bryant ML, Clare M, Houseman KA, Marr JJ, Mueller RA, et al. Getman DP, et al. Among authors: talley jj. J Med Chem. 1993 Jan 22;36(2):288-91. doi: 10.1021/jm00054a014. J Med Chem. 1993. PMID: 8423599 No abstract available.

2

Selective inhibitors of cyclooxygenase-2 (COX-2).

Talley JJ. Talley JJ. Prog Med Chem. 1999;36:201-34. doi: 10.1016/s0079-6468(08)70048-1. Prog Med Chem. 1999. PMID: 10818674 Review. No abstract available.

3

4-[5-Methyl-3-phenylisoxazol-4-yl]- benzenesulfonamide, valdecoxib: a potent and selective inhibitor of COX-2.

Talley JJ, Brown DL, Carter JS, Graneto MJ, Koboldt CM, Masferrer JL, Perkins WE, Rogers RS, Shaffer AF, Zhang YY, Zweifel BS, Seibert K. Talley JJ, et al. J Med Chem. 2000 Mar 9;43(5):775-7. doi: 10.1021/jm990577v. J Med Chem. 2000. PMID: 10715145 No abstract available.

4

Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benze nesulfonamide (SC-58635, celecoxib).

Penning TD, Talley JJ, Bertenshaw SR, Carter JS, Collins PW, Docter S, Graneto MJ, Lee LF, Malecha JW, Miyashiro JM, Rogers RS, Rogier DJ, Yu SS, AndersonGD, Burton EG, Cogburn JN, Gregory SA, Koboldt CM, Perkins WE, Seibert K, Veenhuizen AW, Zhang YY, Isakson PC. Penning TD, et al. Among authors: talley jj. J Med Chem. 1997 Apr 25;40(9):1347-65. doi: 10.1021/jm960803q. J Med Chem. 1997. PMID: 9135032

5

Design and synthesis of sulfonyl-substituted 4,5-diarylthiazoles as selective cyclooxygenase-2 inhibitors.

Carter JS, Rogier DJ, Graneto MJ, Seibert K, Koboldt CM, Zhang Y, Talley JJ. Carter JS, et al. Among authors: talley jj. Bioorg Med Chem Lett. 1999 Apr 19;9(8):1167-70. doi: 10.1016/s0960-894x(99)00158-4. Bioorg Med Chem Lett. 1999. PMID: 10328306

6

Synthesis and activity of sulfonamide-substituted 4,5-diaryl thiazoles as selective cyclooxygenase-2 inhibitors.

Carter JS, Kramer S, Talley JJ, Penning T, Collins P, Graneto MJ, Seibert K, Koboldt CM, Masferrer J, Zweifel B. Carter JS, et al. Among authors: talley jj. Bioorg Med Chem Lett. 1999 Apr 19;9(8):1171-4. doi: 10.1016/s0960-894x(99)00157-2. Bioorg Med Chem Lett. 1999. PMID: 10328307

7

N-[[(5-methyl-3-phenylisoxazol-4-yl)-phenyl]sulfonyl]propanamide, sodium salt, parecoxib sodium: A potent and selective inhibitor of COX-2 for parenteral administration.

Talley JJ, Bertenshaw SR, Brown DL, Carter JS, Graneto MJ, Kellogg MS, Koboldt CM, Yuan J, Zhang YY, Seibert K. Talley JJ, et al. J Med Chem. 2000 May 4;43(9):1661-3. doi: 10.1021/jm000069h. J Med Chem. 2000. PMID: 10794682 No abstract available.

8

Pentafluorosulfanyl-Substituted Benzopyran Analogues As New Cyclooxygenase-2 Inhibitors with Excellent Pharmacokinetics and Efficacy in Blocking Inflammation.

Zhang Y, Wang Y, He C, Liu X, Lu Y, Chen T, Pan Q, Xiong J, She M, Tu Z, Qin X, Li M, Tortorella MD, Talley JJ. Zhang Y, et al. Among authors: talley jj. J Med Chem. 2017 May 25;60(10):4135-4146. doi: 10.1021/acs.jmedchem.6b01484. Epub 2017 May 5. J Med Chem. 2017. PMID: 28475316

9

Synthesis of Deuterated Benzopyran Derivatives as Selective COX-2 Inhibitors with Improved Pharmacokinetic Properties.

Zhang Y, Tortorella MD, Wang Y, Liu J, Tu Z, Liu X, Bai Y, Wen D, Lu X, Lu Y, Talley JJ. Zhang Y, et al. Among authors: talley jj. ACS Med Chem Lett. 2014 Jul 27;5(10):1162-6. doi: 10.1021/ml500299q. eCollection 2014 Oct 9. ACS Med Chem Lett. 2014. PMID: 25313331 Free PMC article.

10

4,5-Diaryloxazole inhibitors of cyclooxygenase-2 (COX-2).

Talley JJ, Bertenshaw SR, Brown DL, Carter JS, Graneto MJ, Koboldt CM, Masferrer JL, Norman BH, Rogier DJ Jr, Zwwifel BS, Seibert K. Talley JJ, et al. Med Res Rev. 1999 May;19(3):199-208. doi: 10.1002/(sici)1098-1128(199905)19:3<199::aid-med1>3.0.co;2-7. Med Res Rev. 1999. PMID: 10232649 Review.

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