Marsh KC - Search Results

1

Azole endothelin antagonists. 3. Using delta log P as a tool to improve absorption.

von Geldern TW, Hoffman DJ, Kester JA, Nellans HN, Dayton BD, Calzadilla SV, Marsh KC, Hernandez L, Chiou W, Dixon DB, Wu-Wong JR, Opgenorth TJ. von Geldern TW, et al. Among authors: marsh kc. J Med Chem. 1996 Feb 16;39(4):982-91. doi: 10.1021/jm9505932. J Med Chem. 1996. PMID: 8632421

2

Synthesis and evaluation of urea-based indazoles as melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity.

Souers AJ, Gao J, Wodka D, Judd AS, Mulhern MM, Napier JJ, Brune ME, Bush EN, Brodjian SJ, Dayton BD, Shapiro R, Hernandez LE, Marsh KC, Sham HL, Collins CA, Kym PR. Souers AJ, et al. Among authors: marsh kc. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2752-7. doi: 10.1016/j.bmcl.2005.03.114. Bioorg Med Chem Lett. 2005. PMID: 15911251

3

Preparation of 9-deoxo-4"-deoxy-6,9-epoxyerythromycin lactams "motilactides": potent and orally active prokinetic agents.

Faghih R, Nellans HN, Lartey PA, Petersen A, Marsh K, Bennani YL, Plattner JJ. Faghih R, et al. Bioorg Med Chem Lett. 1998 Apr 7;8(7):805-10. doi: 10.1016/s0960-894x(98)00111-5. Bioorg Med Chem Lett. 1998. PMID: 9871545

4

2,4-Diarylpyrrolidine-3-carboxylic acids--potent ETA selective endothelin receptor antagonists. 1. Discovery of A-127722.

Winn M, von Geldern TW, Opgenorth TJ, Jae HS, Tasker AS, Boyd SA, Kester JA, Mantei RA, Bal R, Sorensen BK, Wu-Wong JR, Chiou WJ, Dixon DB, Novosad EI, Hernandez L, Marsh KC. Winn M, et al. Among authors: marsh kc. J Med Chem. 1996 Mar 1;39(5):1039-48. doi: 10.1021/jm9505369. J Med Chem. 1996. PMID: 8676339

5

Potent and selective non-benzodioxole-containing endothelin-A receptor antagonists.

Tasker AS, Sorensen BK, Jae HS, Winn M, von Geldern TW, Dixon DB, Chiou WJ, Dayton BD, Calzadila S, Hernandez L, Marsh KC, WuWong JR, Opgenorth TJ. Tasker AS, et al. Among authors: marsh kc. J Med Chem. 1997 Jan 31;40(3):322-30. doi: 10.1021/jm960077r. J Med Chem. 1997. PMID: 9022798

6

Pyrrolidine-3-carboxylic acids as endothelin antagonists. 2. Sulfonamide-based ETA/ETB mixed antagonists.

Jae HS, Winn M, Dixon DB, Marsh KC, Nguyen B, Opgenorth TJ, von Geldern TW. Jae HS, et al. Among authors: marsh kc. J Med Chem. 1997 Sep 26;40(20):3217-27. doi: 10.1021/jm970101g. J Med Chem. 1997. PMID: 9379441

7

Pyrrolidine-3-carboxylic acids as endothelin antagonists. 3. Discovery of a potent, 2-nonaryl, highly selective ETA antagonist (A-216546).

Liu G, Henry KJ Jr, Szczepankiewicz BG, Winn M, Kozmina NS, Boyd SA, Wasicak J, von Geldern TW, Wu-Wong JR, Chiou WJ, Dixon DB, Nguyen B, Marsh KC, Opgenorth TJ. Liu G, et al. Among authors: marsh kc. J Med Chem. 1998 Aug 13;41(17):3261-75. doi: 10.1021/jm980217s. J Med Chem. 1998. PMID: 9703472

8

The effects of diminishing albumin binding to some Endothelin receptor antagonists.

Szczepankiewicz BG, Bal RB, von Geldern TW, Wu-Wong JR, Chiou WJ, Dixon DB, Opgenorth TJ, Hoffman DJ, Borre AJ, Marsh KC, Nguyen BN. Szczepankiewicz BG, et al. Among authors: marsh kc. Life Sci. 1998;63(21):1905-12. doi: 10.1016/s0024-3205(98)00466-4. Life Sci. 1998. PMID: 9825768

9

Discovery of a series of pyrrolidine-based endothelin receptor antagonists with enhanced ET(A) receptor selectivity.

Boyd SA, Mantei RA, Tasker AS, Liu G, Sorensen BK, Henry KJ Jr, von Geldern TW, Winn M, Wu-Wong JR, Chiou WJ, Dixon DB, Hutchins CW, Marsh KC, Nguyen B, Opgenorth TJ. Boyd SA, et al. Among authors: marsh kc. Bioorg Med Chem. 1999 Jun;7(6):991-1002. doi: 10.1016/s0968-0896(99)00022-x. Bioorg Med Chem. 1999. PMID: 10428367

10

Pyrrolidine-3-carboxylic acids as endothelin antagonists. 4. Side chain conformational restriction leads to ET(B) selectivity.

von Geldern TW, Tasker AS, Sorensen BK, Winn M, Szczepankiewicz BG, Dixon DB, Chiou WJ, Wang L, Wessale JL, Adler A, Marsh KC, Nguyen B, Opgenorth TJ. von Geldern TW, et al. Among authors: marsh kc. J Med Chem. 1999 Sep 9;42(18):3668-78. doi: 10.1021/jm990170q. J Med Chem. 1999. PMID: 10479298

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

224 results

Search Page

Filters