Sarau HM - Search Results

1

2-Phenyl-4-quinolinecarboxamides: a novel class of potent and selective non-peptide competitive antagonists for the human neurokinin-3 receptor.

Giardina GA, Sarau HM, Farina C, Medhurst AD, Grugni M, Foley JJ, Raveglia LF, Schmidt DB, Rigolio R, Vassallo M, Vecchietti V, Hay DW. Giardina GA, et al. Among authors: sarau hm. J Med Chem. 1996 Jun 7;39(12):2281-4. doi: 10.1021/jm9602423. J Med Chem. 1996. PMID: 8691422 No abstract available.

2

Synthesis of structural analogs of leukotriene B4 and their receptor binding activity.

Kingsbury WD, Pendrak I, Leber JD, Boehm JC, Mallet B, Sarau HM, Foley JJ, Schmidt DB, Daines RA. Kingsbury WD, et al. Among authors: sarau hm. J Med Chem. 1993 Oct 29;36(22):3308-20. doi: 10.1021/jm00074a012. J Med Chem. 1993. PMID: 8230121

3

Trisubstituted pyridine leukotriene B4 receptor antagonists: synthesis and structure-activity relationships.

Daines RA, Chambers PA, Pendrak I, Jakas DR, Sarau HM, Foley JJ, Schmidt DB, Kingsbury WD. Daines RA, et al. Among authors: sarau hm. J Med Chem. 1993 Oct 29;36(22):3321-32. doi: 10.1021/jm00074a013. J Med Chem. 1993. PMID: 8230122

4

Synthesis and LTB4 receptor antagonist activities of the naturally occurring LTB4 receptor antagonist Leucettamine A and related analogues.

Boehm JC, Gleason JG, Pendrak I, Sarau HM, Schmidt DB, Foley JJ, Kingsbury WD. Boehm JC, et al. Among authors: sarau hm. J Med Chem. 1993 Oct 29;36(22):3333-40. doi: 10.1021/jm00074a014. J Med Chem. 1993. PMID: 8230123

5

(E)-3-[6-[[(2,6-dichlorophenyl)thio]methyl]-3-(2-phenylethoxy)-2- pyridinyl]-2-propenoic acid: a high-affinity leukotriene B4 receptor antagonist with oral antiinflammatory activity.

Daines RA, Chambers PA, Foley JJ, Griswold DE, Kingsbury WD, Martin LD, Schmidt DB, Sham KK, Sarau HM. Daines RA, et al. Among authors: sarau hm. J Med Chem. 1996 Sep 13;39(19):3837-41. doi: 10.1021/jm960248s. J Med Chem. 1996. PMID: 8809171

6

Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.

Sarau HM, Griswold DE, Potts W, Foley JJ, Schmidt DB, Webb EF, Martin LD, Brawner ME, Elshourbagy NA, Medhurst AD, Giardina GA, Hay DW. Sarau HM, et al. J Pharmacol Exp Ther. 1997 Jun;281(3):1303-11. J Pharmacol Exp Ther. 1997. PMID: 9190866

7

Discovery of a novel class of selective non-peptide antagonists for the human neurokinin-3 receptor. 1. Identification of the 4-quinolinecarboxamide framework.

Giardina GA, Sarau HM, Farina C, Medhurst AD, Grugni M, Raveglia LF, Schmidt DB, Rigolio R, Luttmann M, Vecchietti V, Hay DW. Giardina GA, et al. Among authors: sarau hm. J Med Chem. 1997 Jun 6;40(12):1794-807. doi: 10.1021/jm960818o. J Med Chem. 1997. PMID: 9191956

8

Discovery of a novel class of selective non-peptide antagonists for the human neurokinin-3 receptor. 2. Identification of (S)-N-(1-phenylpropyl)-3-hydroxy-2-phenylquinoline-4-carboxamide (SB 223412).

Giardina GA, Raveglia LF, Grugni M, Sarau HM, Farina C, Medhurst AD, Graziani D, Schmidt DB, Rigolio R, Luttmann M, Cavagnera S, Foley JJ, Vecchietti V, Hay DW. Giardina GA, et al. Among authors: sarau hm. J Med Chem. 1999 Mar 25;42(6):1053-65. doi: 10.1021/jm980633c. J Med Chem. 1999. PMID: 10090788

9

Replacement of the quinoline system in 2-phenyl-4-quinolinecarboxamide NK-3 receptor antagonists.

Giardina GA, Artico M, Cavagnera S, Cerri A, Consolandi E, Gagliardi S, Graziani D, Grugni M, Hay DW, Luttmann MA, Mena R, Raveglia LF, Rigolio R, Sarau HM, Schmidt DB, Zanoni G, Farina C. Giardina GA, et al. Among authors: sarau hm. Farmaco. 1999 Jun 30;54(6):364-74. doi: 10.1016/s0014-827x(99)00043-9. Farmaco. 1999. PMID: 10443017

10

Nonpeptide tachykinin receptor antagonists. II. Pharmacological and pharmacokinetic profile of SB-222200, a central nervous system penetrant, potent and selective NK-3 receptor antagonist.

Sarau HM, Griswold DE, Bush B, Potts W, Sandhu P, Lundberg D, Foley JJ, Schmidt DB, Webb EF, Martin LD, Legos JJ, Whitmore RG, Barone FC, Medhurst AD, Luttmann MA, Giardina GA, Hay DW. Sarau HM, et al. J Pharmacol Exp Ther. 2000 Oct;295(1):373-81. J Pharmacol Exp Ther. 2000. PMID: 10992004

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